Inhibitor | Target | Synergistic effect | Radiosensitizer | Reference |
Docetaxel | Microtubules | TMZ | Not tested | 56 |
BI 2536 | PLK1 | TMZ | Yes | 70,71,221 |
BI 6727 | PLK1 | TMZ | Not tested | 71,74 |
GSK461364 | PLK1 | TMZ | Yes | 71,75 |
GW843682X | PLK1 | TMZ | Not tested | 71 |
JNJ-10198409 | PLK1 | Not tested | 70 | |
Abemaciclib | CDK4/6 | TMZ | Not tested | 76,77 |
Dinaciclib | CDK2/CDK5/ CDK1/CDK9 | Not tested | 79 | |
Flavopiridol | CDK1/CDK2/CDK4/CDK6 | TMZ | Not tested | 80-83 |
MK-8776 | CDK2 | Gemcitabine | Not tested | 85 |
ON123300 | CDK4 | Gefitinib | Not tested | 86 |
Palbociclib | CDK4/6 | TMZ ; mTOR inhibitor | Yes | 77,87-90 |
Roscovitine | CDK2/CDK5 | PI3K inhibitor PIK-90 | Not tested | 92,93 |
Alisertib | AURKA | TMZ | Yes | 97-100 |
AZD1152 | AURKA/B | TMZ | Yes | 101,102 |
VX-680 | pan-AURK | Yes | 104 | |
ZM 447439 | AURKA/B | TMZ | Yes | 106 |
YM155 | Survivin | TMZ | Yes | 267 |
M4N | Survivin | TMZ | Yes | 263 |